Display Options:
Small molecule
Approved
OTHER
ORAL
Unknown
Dihydrofolate reductase inhibitor
Small molecule
Approved
Unknown
Unknown
Bacterial Infections; Eye Infections; Infections
Unknown
Small molecule
Unknown
Unknown
Unknown
Colorectal Neoplasms; Intervertebral Disc Degeneration; Respiratory Insufficiency; Head and Neck Neoplasms; Neuralgia; Nutrition Disorders; Opioid-Related Disorders; Pre-Eclampsia; Sinusitis; Spinal Cord Injuries; Toothache; Wounds and Injuries; Back Pain; Diabetic Neuropathies; Genital Neoplasms, Female; Hypospadias; Joint Diseases; Kidney Calculi; Low Back Pain; Neck Pain; Neoplasms; Osteoarthritis; Osteoarthritis, Hip; Osteoarthritis, Knee; Parkinson Disease; Pruritus; Restless Legs Syndrome; Chronic Pain; Pain; Pain, Postoperative; Substance-Related Disorders
Mu opioid receptor agonist
Small molecule
Approved
OTHER
INJECTION; ORAL; RECTAL
Unknown
GABA-A receptor; anion channel positive allosteric modulator
Small molecule
Approved
OTHER
INJECTION; ORAL
Rotator Cuff Injuries; Angioedema; Addison Disease; Adrenal Hyperplasia, Congenital; Anemia, Aplastic; Anemia, Hemolytic; Arthritis, Gouty; Arthritis, Juvenile; Arthritis, Psoriatic; Arthritis, Rheumatoid; Asthma; Bursitis; Dermatitis Herpetiformis; Dermatitis, Atopic; Dermatitis, Contact; Dermatitis, Exfoliative; Dermatitis, Seborrheic; Dermatomyositis; Enteritis; Erythema Multiforme; Eye Diseases; Herpes Zoster Ophthalmicus; Hypercalcemia; Hypersensitivity; Iridocyclitis; Iritis; Leukemia; Lupus Erythematosus, Systemic; Lymphoma; Nephrotic Syndrome; Ophthalmia, Sympathetic; Osteoarthritis; Peptic Ulcer; Pneumonia; Polymyositis; Purpura, Thrombocytopenic, Idiopathic; Stevens-Johnson Syndrome; Synovitis; Tennis Elbow; Tenosynovitis; Thrombocytopenia; Thyroiditis, Subacute; Tuberculosis, Meningeal; Tuberculosis, Pulmonary; Uveitis, Posterior
Glucocorticoid receptor agonist
Small molecule
Approved
Unknown
Unknown
Infections; Loiasis; Elephantiasis, Filarial; Helminthiasis
Unknown
Small molecule
Approved
OTHER
INJECTION; ORAL
Sunburn; Rhinitis, Allergic, Seasonal; Cough; Sinusitis
Histamine H1 receptor antagonist
Small molecule
Approved
OTHER
ORAL
Unknown
Nematode GABA-A receptor positive modulator
Small molecule
Approved
DIABETES DRUGS & ENDOCRINOLOGY; MUSCULOSKELETAL; OTHER; PHARMACOLOGY
ORAL
Low Back Pain; Osteoarthritis, Hip; Osteoarthritis, Knee; Acute Pain; Chronic Pain; Pain; Pain, Postoperative
Mu opioid receptor agonist
Small molecule
Approved
Unknown
Unknown
Pain
Mu opioid receptor agonist
Small molecule
Approved
OTHER
ORAL
Dermatomyositis; Glioblastoma; Graves Ophthalmopathy; Hyperthyroidism; Thyroid Diseases
Thyroid peroxidase inhibitor
Small molecule
Approved
OTHER
INJECTION; ORAL
Irritable Bowel Syndrome
Muscarinic acetylcholine receptor M1 antagonist
Small molecule
Approved
OTHER
INJECTION; OPHTHALMIC; ORAL; OTIC; TOPICAL
Acne Vulgaris; Bacterial Infections; Eye Infections
Bacterial 70S ribosome inhibitor
Small molecule
Approved
OTHER
ORAL
Anemia, Sickle Cell; Digestive System Diseases; Head and Neck Neoplasms; Herpes Simplex; Hypertriglyceridemia; Inflammation; Leukoplakia, Oral; Neuralgia, Postherpetic; Ulcer; Acute Lung Injury; Adenoma; Barrett Esophagus; Blood Coagulation Disorders; Carotid Stenosis; Depressive Disorder, Major; Depressive Disorder, Treatment-Resistant; Disseminated Intravascular Coagulation; Duodenal Ulcer; Endometrial Neoplasms; Glioblastoma; HIV Infections; Heart Diseases; Hypercholesterolemia; Hypertension, Pulmonary; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Lupus Erythematosus, Systemic; Melanoma; Metabolic Syndrome; Nasopharyngeal Neoplasms; Neoplasms; Ovarian Neoplasms; Periodontitis; Placental Insufficiency; Pneumonia, Viral; Pregnancy; Prostatic Neoplasms; Rectal Neoplasms; Respiratory Distress Syndrome; Respiratory Insufficiency; Sepsis; Tension-Type Headache; Tobacco Use Disorder; Tuberculosis; Uterine Cervical Neoplasms; Venous Thrombosis; Vitamin D Deficiency; Abortion, Habitual; Acute Chest Syndrome; Acute Coronary Syndrome; Adenomatous Polyposis Coli; Angina, Stable; Aortic Valve Stenosis; Asthma; Atherosclerosis; Atrial Fibrillation; Bipolar Disorder; Blindness; Brain Infarction; Breast Neoplasms; Carcinoma, Hepatocellular; Carcinoma, Non-Small-Cell Lung; Carcinoma, Squamous Cell; Cardiomyopathy, Hypertrophic; Cardiovascular Diseases; Cataract; Cerebral Infarction; Cerebrovascular Disorders; Colitis, Ulcerative; Colonic Neoplasms; Colorectal Neoplasms; Colorectal Neoplasms, Hereditary Nonpolyposis; Diabetes Mellitus; Diabetes Mellitus, Type 2; Diabetic Retinopathy; Esophageal Neoplasms; Fetal Growth Retardation; Gastrointestinal Hemorrhage; Heart Failure; Hemorrhage; Hypertension; Infertility; Influenza, Human; Intracranial Aneurysm; Intracranial Arteriosclerosis; Ischemia; Ischemic Attack, Transient; Ischemic Stroke; Lipid Metabolism Disorders; Low Back Pain; Macular Degeneration; Meningitis; Mucocutaneous Lymph Node Syndrome; Multiple Myeloma; Multiple Sclerosis; Myocardial Ischemia; Non-ST Elevated Myocardial Infarction; Osteoarthritis; Osteonecrosis; Peptic Ulcer; Peripheral Arterial Disease; Pharyngitis; Pneumonia; Polycythemia Vera; Pre-Eclampsia; Prostatic Neoplasms, Castration-Resistant; Psychotic Disorders; Pulmonary Disease, Chronic Obstructive; Renal Insufficiency, Chronic; Retinal Artery Occlusion; Retinal Vein Occlusion; Rheumatic Heart Disease; ST Elevation Myocardial Infarction; Schizophrenia; Severe Acute Respiratory Syndrome; Stomach Neoplasms; Stomach Ulcer; Thrombocythemia, Essential; Thrombophilia; Varicose Ulcer; Vascular Diseases; Venous Thromboembolism; Wounds and Injuries; Arthritis; Back Pain; Common Cold; Coronary Artery Disease; Dysmenorrhea; Fever; Headache; Migraine Disorders; Muscle Cramp; Myalgia; Myocardial Infarction; Pain; Spasm; Stroke; Thrombosis; Toothache
Cyclooxygenase inhibitor
Small molecule
Approved
Unknown
Unknown
Atrial Fibrillation; Death, Sudden, Cardiac; Heart Failure; Myocardial Infarction; Ventricular Fibrillation; Arrhythmias, Cardiac
Unknown
Small molecule
Approved
OTHER
ORAL
Colitis, Ulcerative; Crohn Disease; Tuberculosis
Dihydrofolate reductase inhibitor
Small molecule
Approved
OTHER
INJECTION; ORAL
Arrhythmias, Cardiac; Malaria
Sodium channel alpha subunit blocker
Small molecule
Approved
Unknown
Unknown
Hepatitis B, Chronic; Rhinitis, Allergic, Seasonal; Sunburn; Influenza, Human; Hypersensitivity
Unknown
Small molecule
Approved
DIABETES DRUGS & ENDOCRINOLOGY; OTHER; RHEUMATOLOGY
ORAL
Glioblastoma; Hypertension, Pulmonary; Intestinal Obstruction; Nausea; Cholangitis, Sclerosing; Peripheral Nervous System Diseases; Spondylitis, Ankylosing; Arthritis, Psoriatic; Arthritis, Juvenile; Arthritis, Rheumatoid; Colitis, Ulcerative
Arachidonate 5-lipoxygenase inhibitor
Small molecule
Approved
Unknown
Unknown
Constipation; Hepatitis B, Chronic; Non-alcoholic Fatty Liver Disease; Respiratory Syncytial Virus Infections; Depressive Disorder; Depressive Disorder, Major; Migraine Disorders; Amyotrophic Lateral Sclerosis; Atrial Fibrillation; Death, Sudden, Cardiac; Multiple Sclerosis; Myocardial Infarction; Ventricular Fibrillation; Arrhythmias, Cardiac
Unknown
Small molecule
Approved
OTHER
INJECTION
Cardiovascular Diseases; Acute Lung Injury; Ischemic Stroke; Hypotension; Poliomyelitis; Sepsis
Adrenergic receptor agonist
Small molecule
Approved
OTHER
OPHTHALMIC
Unknown
Bacterial 70S ribosome inhibitor
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
CARDIOVASCULAR; OTHER
INJECTION; ORAL
Atrial Fibrillation; Heart Failure; Arrhythmias, Cardiac
Sodium channel alpha subunit blocker
Small molecule
Unknown
Unknown
Unknown
Digestive System Diseases
Unknown
Small molecule
Approved
OTHER
ORAL
Epilepsy
Sodium channel alpha subunit blocker
Small molecule
Approved
Unknown
Unknown
Crohn Disease; Gastroparesis; Anxiety; Dementia; Depressive Disorder; Hyperemesis Gravidarum; Migraine with Aura; Migraine without Aura; Nausea; Pain; Schizophrenia; Vertigo; Vomiting; Hypersensitivity; Pruritus
Unknown
Small molecule
Approved
OTHER
ORAL
Amphetamine-Related Disorders; Fatigue; HIV Infections; Multiple Myeloma; Neoplasms; Prostatic Neoplasms, Castration-Resistant; Sarcoma; Alcohol-Related Disorders; Breast Neoplasms; Carcinoma, Non-Small-Cell Lung; Cocaine-Related Disorders; Glioblastoma; Melanoma; Neoplasms, Germ Cell and Embryonal; Opioid-Related Disorders; Pancreatic Neoplasms; Severe Acute Respiratory Syndrome; Alcoholism; Ectoparasitic Infestations
Aldehyde dehydrogenase inhibitor
Small molecule
Approved
Unknown
Unknown
Hypotension, Orthostatic; Orthostatic Intolerance
Unknown
Small molecule
Approved
OTHER
ORAL
Unknown
Unknown
Small molecule
Approved
OTHER
INJECTION
Unknown
Adrenergic receptor agonist
Small molecule
Approved
OTHER
INJECTION
Unknown
Acetylcholinesterase inhibitor
Small molecule
Approved
Unknown
Unknown
Cardiovascular Diseases
Unknown
Small molecule
Approved
OTHER
INJECTION; ORAL
Lung Diseases, Obstructive
Phosphodiesterase 3A inhibitor
Small molecule
Approved
OTHER
ORAL
Unknown
Histamine H2 receptor antagonist
Small molecule
Approved
OTHER
FOR RX COMPOUNDING; INJECTION; OPHTHALMIC; OTIC; RECTAL; TOPICAL
Vitiligo; Dermatitis, Atopic; Eye Diseases; Hemorrhoids; Inflammation; Pruritus; Skin Diseases
Glucocorticoid receptor agonist