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Small molecule
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Hexokinase type IV activator
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Phosphodiesterase isozyme 4 inhibitor
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Prostanoid EP4 receptor agonist
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Serine/threonine-protein kinase Chk1 inhibitor
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G-protein coupled receptor 84 negative allosteric modulator
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Cathepsin S inhibitor
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Voltage-gated calcium channel modulator
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Glutamate receptor ionotropic AMPA antagonist
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Proteinase activated receptor 4 antagonist
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Bromodomain and extra-terminal motif (BET) inhibitor
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Metabotropic glutamate receptor 2 positive allosteric modulator
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Neurokinin 1 receptor antagonist
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Hepatocyte growth factor receptor inhibitor
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Serotonin 4 (5-HT4) receptor agonist
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Mineralocorticoid receptor antagonist
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