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Small molecule
Unknown
Unknown
Investigational
Unknown
Small molecule
Tyrosine-protein kinase TIE-2 inhibitor
Unknown
Investigational
Unknown
Small molecule
Unknown
Unknown
Investigational
Unknown
Small molecule
PI3-kinase p110-delta subunit inhibitor
Unknown
Investigational
Unknown
Small molecule
Calcium-activated potassium channel subunit alpha-1 activator
Unknown
Investigational
Unknown
Small molecule
Isocitrate dehydrogenase [NADP] cytoplasmic inhibitor
Unknown
Investigational
Unknown
Small molecule
Unknown
Unknown
Investigational
Unknown
Small molecule
Neurokinin 3 receptor antagonist
Unknown
Investigational
Unknown
Small molecule
Unknown
Unknown
Investigational
Unknown
Small molecule
Rho-associated protein kinase inhibitor
Unknown
Investigational
Unknown
Small molecule
Unknown
Unknown
Investigational
Unknown
Small molecule
Unknown
Unknown
Investigational
Unknown
Small molecule
Unknown
Unknown
Investigational
Unknown
Small molecule
Tyrosine-protein kinase ABL inhibitor
Unknown
Investigational
Unknown
Small molecule
Tyrosine-protein kinase JAK2 inhibitor
Unknown
Investigational
Unknown
Small molecule
Unknown
Unknown
Investigational
Unknown
Small molecule
Unknown
Unknown
Investigational
Unknown
Small molecule
Unknown
Unknown
Investigational
Unknown
Small molecule
G protein-coupled receptor 44 antagonist
Unknown
Investigational
Unknown
Small molecule
Unknown
Unknown
Investigational
Unknown
Small molecule
Unknown
Unknown
Investigational
Unknown
Small molecule
Unknown
Unknown
Investigational
Unknown
Small molecule
Thymidylate synthase inhibitor
Unknown
Investigational
Unknown
Small molecule
GABA-A receptor; anion channel inverse agonist
Unknown
Investigational
Unknown
Small molecule
Unknown
Unknown
Investigational
Unknown
Small molecule
Unknown
Unknown
Investigational
Unknown
Small molecule
Unknown
Unknown
Investigational
Unknown
Small molecule
Peroxisome proliferator-activated receptor gamma modulator
Unknown
Investigational
Unknown
Small molecule
Unknown
Unknown
Investigational
Unknown
Small molecule
Orexin receptor 1 antagonist
Unknown
Investigational
Unknown
Small molecule
C-C chemokine receptor type 2 antagonist
Unknown
Investigational
Unknown
Small molecule
Unknown
Unknown
Metabolites
Unknown
Small molecule
Unknown
Unknown
Investigational
Unknown
Small molecule
Rho-associated protein kinase inhibitor
Unknown
Investigational
Unknown
Small molecule
Unknown
Unknown
Investigational
Unknown
Small molecule
Muscarinic acetylcholine receptor M1 positive allosteric modulator
Unknown
Investigational
Unknown