Selectivity ratio of pA2 for Cavia porcellus (guinea pig) ileum M3 receptor to pKb for Cavia porcellus (guinea pig) left atria M2 receptor
|
Cavia porcellus
|
13.0
|
|
Selectivity ratio of pA2 for rabbit vas deferens M1 receptor to pKb for guinea pig left atria M2 receptor
|
None
|
35.0
|
|
Selectivity ratio of pKb for rabbit vas deferens M1 receptor to pKb for guinea pig ileum M3 receptor
|
None
|
3.0
|
|
Selectivity ratio of pA2 for rabbit vas deferens M1 receptor to pA2 for guinea pig ileum M3 receptor
|
None
|
3.0
|
|
Antagonist activity at Cavia porcellus (guinea pig) ileum M3 receptor after 30 min
|
Cavia porcellus
|
74.13
nM
|
|
Antagonist activity at Oryctolagus cuniculus (rabbit) vas deferens M1 receptor after 1 hr
|
Oryctolagus cuniculus
|
26.92
nM
|
|
Binding affinity to Cavia porcellus (guinea pig) left atria M2 receptor after 2 hr
|
Cavia porcellus
|
6.02
|
|
Selectivity ratio of pA2 for Cavia porcellus (guinea pig) ileum M3 receptor to pKb for Cavia porcellus (guinea pig) left atria M2 receptor
|
Cavia porcellus
|
13.0
|
|
Selectivity ratio of pA2 for rabbit vas deferens M1 receptor to pKb for guinea pig left atria M2 receptor
|
None
|
35.0
|
|
Binding affinity to Cavia porcellus (guinea pig) left atria M2 receptor after 2 hr
|
Cavia porcellus
|
6.02
|
|
Antagonist activity at Oryctolagus cuniculus (rabbit) vas deferens M1 receptor after 1 hr
|
Oryctolagus cuniculus
|
26.92
nM
|
|
Antagonist activity at Cavia porcellus (guinea pig) ileum M3 receptor after 30 min
|
Cavia porcellus
|
74.13
nM
|
|
Selectivity ratio of pA2 for rabbit vas deferens M1 receptor to pA2 for guinea pig ileum M3 receptor
|
None
|
3.0
|
|