GLPG-0259

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Synonyms
Status
Molecule Category Free-form
UNII 52EG7RFE6Y

Structure

InChI Key YBFGSJUVEOYPIS-OALUTQOASA-N
Smiles CC(C)N1C[C@@H]2C[C@H]1CN2c1ccc(Nc2ncc(-c3coc(C(N)=O)c3)n3ncnc23)cc1
InChI
InChI=1S/C24H26N8O2/c1-14(2)30-10-19-8-18(30)11-31(19)17-5-3-16(4-6-17)29-23-24-27-13-28-32(24)20(9-26-23)15-7-21(22(25)33)34-12-15/h3-7,9,12-14,18-19H,8,10-11H2,1-2H3,(H2,25,33)(H,26,29)/t18-,19-/m0/s1

Pharmacology

Mechanism of Action Action Reference
MAP kinase-activated protein kinase 5 inhibitor INHIBITOR PubMed Other

Target Conservation

Protein: MAP kinase-activated protein kinase 5
Description: MAP kinase-activated protein kinase 5
Organism : Homo sapiens
Q8IW41 ENSG00000089022

Cross References

Resources Reference
ChEMBL CHEMBL3545338
FDA SRS 52EG7RFE6Y
CONTENTS