|
Antifungal activity against Botryotinia fuckeliana at 28 degC after 48 hr microbroth dilution method
|
Botryotinia fuckeliana
|
12.5
ug.mL-1
|
|
Journal : J Agric Food Chem
Title : Metabolites from Aspergillus fumigatus, an endophytic fungus associated with Melia azedarach, and their antifungal, antifeedant, and toxic activities.
Year : 2012
Volume : 60
Issue : 13
First Page : 3424
Last Page : 3431
Authors : Li XJ, Zhang Q, Zhang AL, Gao JM.
Abstract : Thirty-nine fungal metabolites 1-39, including two new alkaloids, 12β-hydroxy-13α-methoxyverruculogen TR-2 (6) and 3-hydroxyfumiquinazoline A (16), were isolated from the fermentation broth of Aspergillus fumigatus LN-4, an endophytic fungus isolated from the stem bark of Melia azedarach. Their structures were elucidated on the basis of detailed spectroscopic analysis (mass spectrometry and one- and two-dimensional NMR experiments) and by comparison of their NMR data with those reported in the literature. These isolated compounds were evaluated for in vitro antifungal activities against some phytopathogenic fungi, toxicity against brine shrimps, and antifeedant activities against armyworm larvae (Mythimna separata Walker). Among them, sixteen compounds showed potent antifungal activities against phytopathogenic fungi (Botrytis cinerea, Alternaria solani, Alternaria alternata, Colletotrichum gloeosporioides, Fusarium solani, Fusarium oxysporum f. sp. niveum, Fusarium oxysporum f. sp. vasinfectum, and Gibberella saubinettii), and four of them, 12β-hydroxy-13α-methoxyverruculogen TR-2 (6), fumitremorgin B (7), verruculogen (8), and helvolic acid (39), exhibited antifungal activities with MIC values of 6.25-50 μg/mL, which were comparable to the two positive controls carbendazim and hymexazol. In addition, of eighteen that exerted moderate lethality toward brine shrimps, compounds 7 and 8 both showed significant toxicities with median lethal concentration (LC(50)) values of 13.6 and 15.8 μg/mL, respectively. Furthermore, among nine metabolites that were found to possess antifeedant activity against armyworm larvae, compounds 7 and 8 gave the best activity with antifeedant indexes (AFI) of 50.0% and 55.0%, respectively. Structure-activity relationships of the metabolites were also discussed.
|
Antifungal activity against Alternaria solani at 28 degC after 48 hr microbroth dilution method
|
Alternaria solani
|
12.5
ug.mL-1
|
|
Journal : J Agric Food Chem
Title : Metabolites from Aspergillus fumigatus, an endophytic fungus associated with Melia azedarach, and their antifungal, antifeedant, and toxic activities.
Year : 2012
Volume : 60
Issue : 13
First Page : 3424
Last Page : 3431
Authors : Li XJ, Zhang Q, Zhang AL, Gao JM.
Abstract : Thirty-nine fungal metabolites 1-39, including two new alkaloids, 12β-hydroxy-13α-methoxyverruculogen TR-2 (6) and 3-hydroxyfumiquinazoline A (16), were isolated from the fermentation broth of Aspergillus fumigatus LN-4, an endophytic fungus isolated from the stem bark of Melia azedarach. Their structures were elucidated on the basis of detailed spectroscopic analysis (mass spectrometry and one- and two-dimensional NMR experiments) and by comparison of their NMR data with those reported in the literature. These isolated compounds were evaluated for in vitro antifungal activities against some phytopathogenic fungi, toxicity against brine shrimps, and antifeedant activities against armyworm larvae (Mythimna separata Walker). Among them, sixteen compounds showed potent antifungal activities against phytopathogenic fungi (Botrytis cinerea, Alternaria solani, Alternaria alternata, Colletotrichum gloeosporioides, Fusarium solani, Fusarium oxysporum f. sp. niveum, Fusarium oxysporum f. sp. vasinfectum, and Gibberella saubinettii), and four of them, 12β-hydroxy-13α-methoxyverruculogen TR-2 (6), fumitremorgin B (7), verruculogen (8), and helvolic acid (39), exhibited antifungal activities with MIC values of 6.25-50 μg/mL, which were comparable to the two positive controls carbendazim and hymexazol. In addition, of eighteen that exerted moderate lethality toward brine shrimps, compounds 7 and 8 both showed significant toxicities with median lethal concentration (LC(50)) values of 13.6 and 15.8 μg/mL, respectively. Furthermore, among nine metabolites that were found to possess antifeedant activity against armyworm larvae, compounds 7 and 8 gave the best activity with antifeedant indexes (AFI) of 50.0% and 55.0%, respectively. Structure-activity relationships of the metabolites were also discussed.
|
Antifungal activity against Alternaria alternata at 28 degC after 48 hr microbroth dilution method
|
Alternaria alternata
|
12.5
ug.mL-1
|
|
Journal : J Agric Food Chem
Title : Metabolites from Aspergillus fumigatus, an endophytic fungus associated with Melia azedarach, and their antifungal, antifeedant, and toxic activities.
Year : 2012
Volume : 60
Issue : 13
First Page : 3424
Last Page : 3431
Authors : Li XJ, Zhang Q, Zhang AL, Gao JM.
Abstract : Thirty-nine fungal metabolites 1-39, including two new alkaloids, 12β-hydroxy-13α-methoxyverruculogen TR-2 (6) and 3-hydroxyfumiquinazoline A (16), were isolated from the fermentation broth of Aspergillus fumigatus LN-4, an endophytic fungus isolated from the stem bark of Melia azedarach. Their structures were elucidated on the basis of detailed spectroscopic analysis (mass spectrometry and one- and two-dimensional NMR experiments) and by comparison of their NMR data with those reported in the literature. These isolated compounds were evaluated for in vitro antifungal activities against some phytopathogenic fungi, toxicity against brine shrimps, and antifeedant activities against armyworm larvae (Mythimna separata Walker). Among them, sixteen compounds showed potent antifungal activities against phytopathogenic fungi (Botrytis cinerea, Alternaria solani, Alternaria alternata, Colletotrichum gloeosporioides, Fusarium solani, Fusarium oxysporum f. sp. niveum, Fusarium oxysporum f. sp. vasinfectum, and Gibberella saubinettii), and four of them, 12β-hydroxy-13α-methoxyverruculogen TR-2 (6), fumitremorgin B (7), verruculogen (8), and helvolic acid (39), exhibited antifungal activities with MIC values of 6.25-50 μg/mL, which were comparable to the two positive controls carbendazim and hymexazol. In addition, of eighteen that exerted moderate lethality toward brine shrimps, compounds 7 and 8 both showed significant toxicities with median lethal concentration (LC(50)) values of 13.6 and 15.8 μg/mL, respectively. Furthermore, among nine metabolites that were found to possess antifeedant activity against armyworm larvae, compounds 7 and 8 gave the best activity with antifeedant indexes (AFI) of 50.0% and 55.0%, respectively. Structure-activity relationships of the metabolites were also discussed.
|
Antifungal activity against Colletotrichum gloeosporioides at 28 degC after 48 hr microbroth dilution method
|
Colletotrichum gloeosporioides
|
12.5
ug.mL-1
|
|
Journal : J Agric Food Chem
Title : Metabolites from Aspergillus fumigatus, an endophytic fungus associated with Melia azedarach, and their antifungal, antifeedant, and toxic activities.
Year : 2012
Volume : 60
Issue : 13
First Page : 3424
Last Page : 3431
Authors : Li XJ, Zhang Q, Zhang AL, Gao JM.
Abstract : Thirty-nine fungal metabolites 1-39, including two new alkaloids, 12β-hydroxy-13α-methoxyverruculogen TR-2 (6) and 3-hydroxyfumiquinazoline A (16), were isolated from the fermentation broth of Aspergillus fumigatus LN-4, an endophytic fungus isolated from the stem bark of Melia azedarach. Their structures were elucidated on the basis of detailed spectroscopic analysis (mass spectrometry and one- and two-dimensional NMR experiments) and by comparison of their NMR data with those reported in the literature. These isolated compounds were evaluated for in vitro antifungal activities against some phytopathogenic fungi, toxicity against brine shrimps, and antifeedant activities against armyworm larvae (Mythimna separata Walker). Among them, sixteen compounds showed potent antifungal activities against phytopathogenic fungi (Botrytis cinerea, Alternaria solani, Alternaria alternata, Colletotrichum gloeosporioides, Fusarium solani, Fusarium oxysporum f. sp. niveum, Fusarium oxysporum f. sp. vasinfectum, and Gibberella saubinettii), and four of them, 12β-hydroxy-13α-methoxyverruculogen TR-2 (6), fumitremorgin B (7), verruculogen (8), and helvolic acid (39), exhibited antifungal activities with MIC values of 6.25-50 μg/mL, which were comparable to the two positive controls carbendazim and hymexazol. In addition, of eighteen that exerted moderate lethality toward brine shrimps, compounds 7 and 8 both showed significant toxicities with median lethal concentration (LC(50)) values of 13.6 and 15.8 μg/mL, respectively. Furthermore, among nine metabolites that were found to possess antifeedant activity against armyworm larvae, compounds 7 and 8 gave the best activity with antifeedant indexes (AFI) of 50.0% and 55.0%, respectively. Structure-activity relationships of the metabolites were also discussed.
|
Antifungal activity against Fusarium solani at 28 degC after 48 hr microbroth dilution method
|
Fusarium solani
|
50.0
ug.mL-1
|
|
Journal : J Agric Food Chem
Title : Metabolites from Aspergillus fumigatus, an endophytic fungus associated with Melia azedarach, and their antifungal, antifeedant, and toxic activities.
Year : 2012
Volume : 60
Issue : 13
First Page : 3424
Last Page : 3431
Authors : Li XJ, Zhang Q, Zhang AL, Gao JM.
Abstract : Thirty-nine fungal metabolites 1-39, including two new alkaloids, 12β-hydroxy-13α-methoxyverruculogen TR-2 (6) and 3-hydroxyfumiquinazoline A (16), were isolated from the fermentation broth of Aspergillus fumigatus LN-4, an endophytic fungus isolated from the stem bark of Melia azedarach. Their structures were elucidated on the basis of detailed spectroscopic analysis (mass spectrometry and one- and two-dimensional NMR experiments) and by comparison of their NMR data with those reported in the literature. These isolated compounds were evaluated for in vitro antifungal activities against some phytopathogenic fungi, toxicity against brine shrimps, and antifeedant activities against armyworm larvae (Mythimna separata Walker). Among them, sixteen compounds showed potent antifungal activities against phytopathogenic fungi (Botrytis cinerea, Alternaria solani, Alternaria alternata, Colletotrichum gloeosporioides, Fusarium solani, Fusarium oxysporum f. sp. niveum, Fusarium oxysporum f. sp. vasinfectum, and Gibberella saubinettii), and four of them, 12β-hydroxy-13α-methoxyverruculogen TR-2 (6), fumitremorgin B (7), verruculogen (8), and helvolic acid (39), exhibited antifungal activities with MIC values of 6.25-50 μg/mL, which were comparable to the two positive controls carbendazim and hymexazol. In addition, of eighteen that exerted moderate lethality toward brine shrimps, compounds 7 and 8 both showed significant toxicities with median lethal concentration (LC(50)) values of 13.6 and 15.8 μg/mL, respectively. Furthermore, among nine metabolites that were found to possess antifeedant activity against armyworm larvae, compounds 7 and 8 gave the best activity with antifeedant indexes (AFI) of 50.0% and 55.0%, respectively. Structure-activity relationships of the metabolites were also discussed.
|
Antifungal activity against Fusarium oxysporum f. sp. niveum at 28 degC after 48 hr microbroth dilution method
|
Fusarium oxysporum f. sp. niveum
|
12.5
ug.mL-1
|
|
Journal : J Agric Food Chem
Title : Metabolites from Aspergillus fumigatus, an endophytic fungus associated with Melia azedarach, and their antifungal, antifeedant, and toxic activities.
Year : 2012
Volume : 60
Issue : 13
First Page : 3424
Last Page : 3431
Authors : Li XJ, Zhang Q, Zhang AL, Gao JM.
Abstract : Thirty-nine fungal metabolites 1-39, including two new alkaloids, 12β-hydroxy-13α-methoxyverruculogen TR-2 (6) and 3-hydroxyfumiquinazoline A (16), were isolated from the fermentation broth of Aspergillus fumigatus LN-4, an endophytic fungus isolated from the stem bark of Melia azedarach. Their structures were elucidated on the basis of detailed spectroscopic analysis (mass spectrometry and one- and two-dimensional NMR experiments) and by comparison of their NMR data with those reported in the literature. These isolated compounds were evaluated for in vitro antifungal activities against some phytopathogenic fungi, toxicity against brine shrimps, and antifeedant activities against armyworm larvae (Mythimna separata Walker). Among them, sixteen compounds showed potent antifungal activities against phytopathogenic fungi (Botrytis cinerea, Alternaria solani, Alternaria alternata, Colletotrichum gloeosporioides, Fusarium solani, Fusarium oxysporum f. sp. niveum, Fusarium oxysporum f. sp. vasinfectum, and Gibberella saubinettii), and four of them, 12β-hydroxy-13α-methoxyverruculogen TR-2 (6), fumitremorgin B (7), verruculogen (8), and helvolic acid (39), exhibited antifungal activities with MIC values of 6.25-50 μg/mL, which were comparable to the two positive controls carbendazim and hymexazol. In addition, of eighteen that exerted moderate lethality toward brine shrimps, compounds 7 and 8 both showed significant toxicities with median lethal concentration (LC(50)) values of 13.6 and 15.8 μg/mL, respectively. Furthermore, among nine metabolites that were found to possess antifeedant activity against armyworm larvae, compounds 7 and 8 gave the best activity with antifeedant indexes (AFI) of 50.0% and 55.0%, respectively. Structure-activity relationships of the metabolites were also discussed.
|
Antifungal activity against Fusarium oxysporum f. sp. vasinfectum at 28 degC after 48 hr microbroth dilution method
|
Fusarium oxysporum f. sp. vasinfectum
|
25.0
ug.mL-1
|
|
Journal : J Agric Food Chem
Title : Metabolites from Aspergillus fumigatus, an endophytic fungus associated with Melia azedarach, and their antifungal, antifeedant, and toxic activities.
Year : 2012
Volume : 60
Issue : 13
First Page : 3424
Last Page : 3431
Authors : Li XJ, Zhang Q, Zhang AL, Gao JM.
Abstract : Thirty-nine fungal metabolites 1-39, including two new alkaloids, 12β-hydroxy-13α-methoxyverruculogen TR-2 (6) and 3-hydroxyfumiquinazoline A (16), were isolated from the fermentation broth of Aspergillus fumigatus LN-4, an endophytic fungus isolated from the stem bark of Melia azedarach. Their structures were elucidated on the basis of detailed spectroscopic analysis (mass spectrometry and one- and two-dimensional NMR experiments) and by comparison of their NMR data with those reported in the literature. These isolated compounds were evaluated for in vitro antifungal activities against some phytopathogenic fungi, toxicity against brine shrimps, and antifeedant activities against armyworm larvae (Mythimna separata Walker). Among them, sixteen compounds showed potent antifungal activities against phytopathogenic fungi (Botrytis cinerea, Alternaria solani, Alternaria alternata, Colletotrichum gloeosporioides, Fusarium solani, Fusarium oxysporum f. sp. niveum, Fusarium oxysporum f. sp. vasinfectum, and Gibberella saubinettii), and four of them, 12β-hydroxy-13α-methoxyverruculogen TR-2 (6), fumitremorgin B (7), verruculogen (8), and helvolic acid (39), exhibited antifungal activities with MIC values of 6.25-50 μg/mL, which were comparable to the two positive controls carbendazim and hymexazol. In addition, of eighteen that exerted moderate lethality toward brine shrimps, compounds 7 and 8 both showed significant toxicities with median lethal concentration (LC(50)) values of 13.6 and 15.8 μg/mL, respectively. Furthermore, among nine metabolites that were found to possess antifeedant activity against armyworm larvae, compounds 7 and 8 gave the best activity with antifeedant indexes (AFI) of 50.0% and 55.0%, respectively. Structure-activity relationships of the metabolites were also discussed.
|
Antifungal activity against Fusarium graminearum at 28 degC after 48 hr microbroth dilution method
|
Fusarium graminearum
|
12.5
ug.mL-1
|
|
Journal : J Agric Food Chem
Title : Metabolites from Aspergillus fumigatus, an endophytic fungus associated with Melia azedarach, and their antifungal, antifeedant, and toxic activities.
Year : 2012
Volume : 60
Issue : 13
First Page : 3424
Last Page : 3431
Authors : Li XJ, Zhang Q, Zhang AL, Gao JM.
Abstract : Thirty-nine fungal metabolites 1-39, including two new alkaloids, 12β-hydroxy-13α-methoxyverruculogen TR-2 (6) and 3-hydroxyfumiquinazoline A (16), were isolated from the fermentation broth of Aspergillus fumigatus LN-4, an endophytic fungus isolated from the stem bark of Melia azedarach. Their structures were elucidated on the basis of detailed spectroscopic analysis (mass spectrometry and one- and two-dimensional NMR experiments) and by comparison of their NMR data with those reported in the literature. These isolated compounds were evaluated for in vitro antifungal activities against some phytopathogenic fungi, toxicity against brine shrimps, and antifeedant activities against armyworm larvae (Mythimna separata Walker). Among them, sixteen compounds showed potent antifungal activities against phytopathogenic fungi (Botrytis cinerea, Alternaria solani, Alternaria alternata, Colletotrichum gloeosporioides, Fusarium solani, Fusarium oxysporum f. sp. niveum, Fusarium oxysporum f. sp. vasinfectum, and Gibberella saubinettii), and four of them, 12β-hydroxy-13α-methoxyverruculogen TR-2 (6), fumitremorgin B (7), verruculogen (8), and helvolic acid (39), exhibited antifungal activities with MIC values of 6.25-50 μg/mL, which were comparable to the two positive controls carbendazim and hymexazol. In addition, of eighteen that exerted moderate lethality toward brine shrimps, compounds 7 and 8 both showed significant toxicities with median lethal concentration (LC(50)) values of 13.6 and 15.8 μg/mL, respectively. Furthermore, among nine metabolites that were found to possess antifeedant activity against armyworm larvae, compounds 7 and 8 gave the best activity with antifeedant indexes (AFI) of 50.0% and 55.0%, respectively. Structure-activity relationships of the metabolites were also discussed.
|
Antifungal activity against Cytospora mandshurica assessed as mycelial growth inhibition
|
Cytospora
|
39.26
ug.mL-1
|
|
Journal : Molecules
Year : 2011
Volume : 16
Issue : 11
First Page : 9129
Last Page : 9141
|
Antifungal activity against Fusarium oxysporum assessed as mycelial growth inhibition
|
Fusarium oxysporum
|
27.93
ug.mL-1
|
|
Journal : Molecules
Year : 2011
Volume : 16
Issue : 11
First Page : 9129
Last Page : 9141
|
Antifungal activity against Thanatephorus cucumeris assessed as mycelial growth inhibition
|
Thanatephorus cucumeris
|
32.21
ug.mL-1
|
|
Journal : Molecules
Year : 2011
Volume : 16
Issue : 11
First Page : 9129
Last Page : 9141
|
Antifungal activity against Sclerotinia sclerotiorum assessed as mycelial growth inhibition
|
Sclerotinia sclerotiorum
|
7.76
ug.mL-1
|
|
Journal : Molecules
Year : 2011
Volume : 16
Issue : 11
First Page : 9129
Last Page : 9141
|
Antifungal activity against Colletotrichum gloeosporioides assessed as mycelial growth inhibition
|
Colletotrichum gloeosporioides
|
37.58
ug.mL-1
|
|
Journal : Molecules
Year : 2011
Volume : 16
Issue : 11
First Page : 9129
Last Page : 9141
|
Antifungal activity against Phytophthora infestans assessed as mycelial growth inhibition
|
Phytophthora infestans
|
26.49
ug.mL-1
|
|
Journal : Molecules
Year : 2011
Volume : 16
Issue : 11
First Page : 9129
Last Page : 9141
|
Antifungal activity against Botryotinia fuckeliana assessed as mycelial growth inhibition
|
Botryotinia fuckeliana
|
25.23
ug.mL-1
|
|
Journal : Molecules
Year : 2011
Volume : 16
Issue : 11
First Page : 9129
Last Page : 9141
|
Antifungal activity against Rhizoctonia solani assessed as mycelial growth inhibition
|
Rhizoctonia solani
|
38.64
ug.mL-1
|
|
Journal : Molecules
Year : 2011
Volume : 16
Issue : 11
First Page : 9129
Last Page : 9141
|
Antifungal activity against Cytospora mandshurica at 50 ug/ml after 5 days by poison plate technique
|
Cytospora
|
57.3
%
|
|
Journal : Molecules
Year : 2011
Volume : 16
Issue : 11
First Page : 9129
Last Page : 9141
|
Antifungal activity against Fusarium oxysporum at 50 ug/ml after 5 days by poison plate technique
|
Fusarium oxysporum
|
58.4
%
|
|
Journal : Molecules
Year : 2011
Volume : 16
Issue : 11
First Page : 9129
Last Page : 9141
|
Antifungal activity against Thanatephorus cucumeris at 50 ug/ml by poisoned food technique
|
Thanatephorus cucumeris
|
78.4
%
|
|
Journal : Molecules
Title : Synthesis and Antifungal Activities of Some Novel Pyrimidine Derivatives
Year : 2011
Volume : 16
Issue : 7
First Page : 5618
Last Page : 5628
Authors : Sun L, Wu J, Zhang L, Luo M, Sun D.
Abstract : Three series of new pyrimidine derivatives were synthesized and their antifungal activities were evaluated in vitro against fourteen phytopathogenic fungi. The results indicated that most of the synthesized compounds possessed fungicidal activities and some of them are more potent than the control fungicides. Preliminary SAR was also discussed.
|
Antifungal activity against Sclerotinia sclerotiorum at 50 ug/ml by poisoned food technique
|
Sclerotinia sclerotiorum
|
66.7
%
|
|
Journal : Molecules
Title : Synthesis and Antifungal Activities of Some Novel Pyrimidine Derivatives
Year : 2011
Volume : 16
Issue : 7
First Page : 5618
Last Page : 5628
Authors : Sun L, Wu J, Zhang L, Luo M, Sun D.
Abstract : Three series of new pyrimidine derivatives were synthesized and their antifungal activities were evaluated in vitro against fourteen phytopathogenic fungi. The results indicated that most of the synthesized compounds possessed fungicidal activities and some of them are more potent than the control fungicides. Preliminary SAR was also discussed.
|
Antifungal activity against Ceratobasidium cereale at 50 ug/ml by poisoned food technique
|
Ceratobasidium cereale
|
25.0
%
|
|
Journal : Molecules
Title : Synthesis and Antifungal Activities of Some Novel Pyrimidine Derivatives
Year : 2011
Volume : 16
Issue : 7
First Page : 5618
Last Page : 5628
Authors : Sun L, Wu J, Zhang L, Luo M, Sun D.
Abstract : Three series of new pyrimidine derivatives were synthesized and their antifungal activities were evaluated in vitro against fourteen phytopathogenic fungi. The results indicated that most of the synthesized compounds possessed fungicidal activities and some of them are more potent than the control fungicides. Preliminary SAR was also discussed.
|
Antifungal activity against Rhizoctonia solani at 50 ug/ml by poisoned food technique
|
Rhizoctonia solani
|
63.5
%
|
|
Journal : Molecules
Title : Synthesis and Antifungal Activities of Some Novel Pyrimidine Derivatives
Year : 2011
Volume : 16
Issue : 7
First Page : 5618
Last Page : 5628
Authors : Sun L, Wu J, Zhang L, Luo M, Sun D.
Abstract : Three series of new pyrimidine derivatives were synthesized and their antifungal activities were evaluated in vitro against fourteen phytopathogenic fungi. The results indicated that most of the synthesized compounds possessed fungicidal activities and some of them are more potent than the control fungicides. Preliminary SAR was also discussed.
|
Antifungal activity against Phytophthora infestans at 50 ug/ml by poisoned food technique
|
Phytophthora infestans
|
36.4
%
|
|
Journal : Molecules
Title : Synthesis and Antifungal Activities of Some Novel Pyrimidine Derivatives
Year : 2011
Volume : 16
Issue : 7
First Page : 5618
Last Page : 5628
Authors : Sun L, Wu J, Zhang L, Luo M, Sun D.
Abstract : Three series of new pyrimidine derivatives were synthesized and their antifungal activities were evaluated in vitro against fourteen phytopathogenic fungi. The results indicated that most of the synthesized compounds possessed fungicidal activities and some of them are more potent than the control fungicides. Preliminary SAR was also discussed.
|
Antifungal activity against Macrophoma kuwatsukai at 50 ug/ml by poisoned food technique
|
Macrophoma
|
50.0
%
|
|
Journal : Molecules
Title : Synthesis and Antifungal Activities of Some Novel Pyrimidine Derivatives
Year : 2011
Volume : 16
Issue : 7
First Page : 5618
Last Page : 5628
Authors : Sun L, Wu J, Zhang L, Luo M, Sun D.
Abstract : Three series of new pyrimidine derivatives were synthesized and their antifungal activities were evaluated in vitro against fourteen phytopathogenic fungi. The results indicated that most of the synthesized compounds possessed fungicidal activities and some of them are more potent than the control fungicides. Preliminary SAR was also discussed.
|
Antifungal activity against Fusarium fujikuroi at 50 ug/ml by poisoned food technique
|
Fusarium fujikuroi
|
40.0
%
|
|
Journal : Molecules
Title : Synthesis and Antifungal Activities of Some Novel Pyrimidine Derivatives
Year : 2011
Volume : 16
Issue : 7
First Page : 5618
Last Page : 5628
Authors : Sun L, Wu J, Zhang L, Luo M, Sun D.
Abstract : Three series of new pyrimidine derivatives were synthesized and their antifungal activities were evaluated in vitro against fourteen phytopathogenic fungi. The results indicated that most of the synthesized compounds possessed fungicidal activities and some of them are more potent than the control fungicides. Preliminary SAR was also discussed.
|
Antifungal activity against Fusarium graminearum at 50 ug/ml by poisoned food technique
|
Fusarium graminearum
|
33.3
%
|
|
Journal : Molecules
Title : Synthesis and Antifungal Activities of Some Novel Pyrimidine Derivatives
Year : 2011
Volume : 16
Issue : 7
First Page : 5618
Last Page : 5628
Authors : Sun L, Wu J, Zhang L, Luo M, Sun D.
Abstract : Three series of new pyrimidine derivatives were synthesized and their antifungal activities were evaluated in vitro against fourteen phytopathogenic fungi. The results indicated that most of the synthesized compounds possessed fungicidal activities and some of them are more potent than the control fungicides. Preliminary SAR was also discussed.
|
Antifungal activity against Mycosphaerella arachidis at 50 ug/ml by poisoned food technique
|
Mycosphaerella arachidis
|
93.3
%
|
|
Journal : Molecules
Title : Synthesis and Antifungal Activities of Some Novel Pyrimidine Derivatives
Year : 2011
Volume : 16
Issue : 7
First Page : 5618
Last Page : 5628
Authors : Sun L, Wu J, Zhang L, Luo M, Sun D.
Abstract : Three series of new pyrimidine derivatives were synthesized and their antifungal activities were evaluated in vitro against fourteen phytopathogenic fungi. The results indicated that most of the synthesized compounds possessed fungicidal activities and some of them are more potent than the control fungicides. Preliminary SAR was also discussed.
|
Antifungal activity against Cochliobolus heterostrophus at 50 ug/ml by poisoned food technique
|
Cochliobolus heterostrophus
|
34.8
%
|
|
Journal : Molecules
Title : Synthesis and Antifungal Activities of Some Novel Pyrimidine Derivatives
Year : 2011
Volume : 16
Issue : 7
First Page : 5618
Last Page : 5628
Authors : Sun L, Wu J, Zhang L, Luo M, Sun D.
Abstract : Three series of new pyrimidine derivatives were synthesized and their antifungal activities were evaluated in vitro against fourteen phytopathogenic fungi. The results indicated that most of the synthesized compounds possessed fungicidal activities and some of them are more potent than the control fungicides. Preliminary SAR was also discussed.
|
Antifungal activity against Botryotinia fuckeliana at 50 ug/ml by poisoned food technique
|
Botryotinia fuckeliana
|
70.4
%
|
|
Journal : Molecules
Title : Synthesis and Antifungal Activities of Some Novel Pyrimidine Derivatives
Year : 2011
Volume : 16
Issue : 7
First Page : 5618
Last Page : 5628
Authors : Sun L, Wu J, Zhang L, Luo M, Sun D.
Abstract : Three series of new pyrimidine derivatives were synthesized and their antifungal activities were evaluated in vitro against fourteen phytopathogenic fungi. The results indicated that most of the synthesized compounds possessed fungicidal activities and some of them are more potent than the control fungicides. Preliminary SAR was also discussed.
|
Antifungal activity against Alternaria solani at 50 ug/ml by poisoned food technique
|
Alternaria solani
|
88.2
%
|
|
Journal : Molecules
Title : Synthesis and Antifungal Activities of Some Novel Pyrimidine Derivatives
Year : 2011
Volume : 16
Issue : 7
First Page : 5618
Last Page : 5628
Authors : Sun L, Wu J, Zhang L, Luo M, Sun D.
Abstract : Three series of new pyrimidine derivatives were synthesized and their antifungal activities were evaluated in vitro against fourteen phytopathogenic fungi. The results indicated that most of the synthesized compounds possessed fungicidal activities and some of them are more potent than the control fungicides. Preliminary SAR was also discussed.
|
Antifungal activity against Alternaria mali at 50 ug/ml by poisoned food technique
|
Alternaria mali
|
85.7
%
|
|
Journal : Molecules
Title : Synthesis and Antifungal Activities of Some Novel Pyrimidine Derivatives
Year : 2011
Volume : 16
Issue : 7
First Page : 5618
Last Page : 5628
Authors : Sun L, Wu J, Zhang L, Luo M, Sun D.
Abstract : Three series of new pyrimidine derivatives were synthesized and their antifungal activities were evaluated in vitro against fourteen phytopathogenic fungi. The results indicated that most of the synthesized compounds possessed fungicidal activities and some of them are more potent than the control fungicides. Preliminary SAR was also discussed.
|
Antifungal activity against Alternaria kikuchiana at 50 ug/ml by poisoned food technique
|
Alternaria kikuchiana
|
81.8
%
|
|
Journal : Molecules
Title : Synthesis and Antifungal Activities of Some Novel Pyrimidine Derivatives
Year : 2011
Volume : 16
Issue : 7
First Page : 5618
Last Page : 5628
Authors : Sun L, Wu J, Zhang L, Luo M, Sun D.
Abstract : Three series of new pyrimidine derivatives were synthesized and their antifungal activities were evaluated in vitro against fourteen phytopathogenic fungi. The results indicated that most of the synthesized compounds possessed fungicidal activities and some of them are more potent than the control fungicides. Preliminary SAR was also discussed.
|
Fungicidal activity against Alternaria alternata APS-38 assessed as mycelial growth inhibition at 25 mg/L after 3 days
|
Alternaria alternata
|
74.0
%
|
|
Journal : J Pesticide Sci
Year : 2012
Volume : 37
Issue : 1
First Page : 89
Last Page : 94
|
Fungicidal activity against Gaeumannomyces graminis MAFF305168 assessed as mycelial growth inhibition at 25 mg/L after 1 day
|
Gaeumannomyces graminis
|
56.0
%
|
|
Journal : J Pesticide Sci
Year : 2012
Volume : 37
Issue : 1
First Page : 89
Last Page : 94
|
Fungicidal activity against Rhizoctonia solani ET0007 assessed as mycelial growth inhibition at 25 mg/L after 1 day
|
Rhizoctonia solani
|
28.0
%
|
|
Journal : J Pesticide Sci
Year : 2012
Volume : 37
Issue : 1
First Page : 89
Last Page : 94
|
Fungicidal activity against Microdochium nivale IFO-7432 assessed as mycelial growth inhibition at 25 mg/L after 3 days
|
Microdochium nivale
|
77.0
%
|
|
Journal : J Pesticide Sci
Year : 2012
Volume : 37
Issue : 1
First Page : 89
Last Page : 94
|
Fungicidal activity against Zymoseptoria tritici S3 assessed as mycelial growth inhibition at 25 mg/L after 14 days
|
Zymoseptoria tritici
|
86.0
%
|
|
Journal : J Pesticide Sci
Year : 2012
Volume : 37
Issue : 1
First Page : 89
Last Page : 94
|
Fungicidal activity against Rhynchosporium secalis IFO-5290 assessed as mycelial growth inhibition at 25 mg/L after 14 days
|
Rhynchosporium secalis
|
100.0
%
|
|
Journal : J Pesticide Sci
Year : 2012
Volume : 37
Issue : 1
First Page : 89
Last Page : 94
|
Fungicidal activity against Cercospora beticola Be-2-6 assessed as mycelial growth inhibition at 25 mg/L after 7 days
|
Cercospora beticola
|
88.0
%
|
|
Journal : J Pesticide Sci
Year : 2012
Volume : 37
Issue : 1
First Page : 89
Last Page : 94
|
Fungicidal activity against Fusarium graminearum H3 assessed as mycelial growth inhibition at 25 mg/L after 3 days
|
Fusarium graminearum
|
45.0
%
|
|
Journal : J Pesticide Sci
Year : 2012
Volume : 37
Issue : 1
First Page : 89
Last Page : 94
|
Fungicidal activity against Pyrenophora graminea IFO-7507 assessed as mycelial growth inhibition at 25 mg/L after 3 days
|
Pyrenophora graminea
|
80.0
%
|
|
Journal : J Pesticide Sci
Year : 2012
Volume : 37
Issue : 1
First Page : 89
Last Page : 94
|
Growth inhibition of Bipolaris sorokiniana at 50 ug/ml after 4 days by poisoned food technique
|
Bipolaris sorokiniana
|
100.0
%
|
|
Journal : Chem Pharm Bull (Tokyo)
Year : 2007
Volume : 55
Issue : 12
First Page : 1755
Last Page : 1757
|
Growth inhibition of Bipolaris sorokiniana at 500 ug/ml after 4 days by poisoned food technique
|
Bipolaris sorokiniana
|
37.1
%
|
|
Journal : Chem Pharm Bull (Tokyo)
Year : 2007
Volume : 55
Issue : 12
First Page : 1755
Last Page : 1757
|
Growth inhibition of Alternaria brassicae at 50 ug/ml after 4 days by poisoned food technique
|
Alternaria brassicae
|
89.0
%
|
|
Journal : Chem Pharm Bull (Tokyo)
Year : 2007
Volume : 55
Issue : 12
First Page : 1755
Last Page : 1757
|
Growth inhibition of Alternaria brassicae at 500 ug/ml after 4 days by poisoned food technique
|
Alternaria brassicae
|
100.0
%
|
|
Journal : Chem Pharm Bull (Tokyo)
Year : 2007
Volume : 55
Issue : 12
First Page : 1755
Last Page : 1757
|
Growth inhibition of Fusarium oxysporum f. sp. cucumerinum at 50 ug/ml after 4 days by poisoned food technique
|
Fusarium oxysporum f. sp. cucumerinum
|
19.8
%
|
|
Journal : Chem Pharm Bull (Tokyo)
Year : 2007
Volume : 55
Issue : 12
First Page : 1755
Last Page : 1757
|
Growth inhibition of Fusarium oxysporum f. sp. cucumerinum at 500 ug/ml after 4 days by poisoned food technique
|
Fusarium oxysporum f. sp. cucumerinum
|
91.5
%
|
|
Journal : Chem Pharm Bull (Tokyo)
Year : 2007
Volume : 55
Issue : 12
First Page : 1755
Last Page : 1757
|
Growth inhibition of Fusarium oxysporum f. sp. vasinfectum at 50 ug/ml after 4 days by poisoned food technique
|
Fusarium oxysporum f. sp. vasinfectum
|
45.8
%
|
|
Journal : Chem Pharm Bull (Tokyo)
Year : 2007
Volume : 55
Issue : 12
First Page : 1755
Last Page : 1757
|
Growth inhibition of Fusarium oxysporum f. sp. vasinfectum at 500 ug/ml after 4 days by poisoned food technique
|
Fusarium oxysporum f. sp. vasinfectum
|
92.3
%
|
|
Journal : Chem Pharm Bull (Tokyo)
Year : 2007
Volume : 55
Issue : 12
First Page : 1755
Last Page : 1757
|
Growth inhibition of Magnaporthe oryzae at 50 ug/ml after 4 days by poisoned food technique
|
Magnaporthe oryzae
|
66.4
%
|
|
Journal : Chem Pharm Bull (Tokyo)
Year : 2007
Volume : 55
Issue : 12
First Page : 1755
Last Page : 1757
|
Growth inhibition of Magnaporthe oryzae at 500 ug/ml after 4 days by poisoned food technique
|
Magnaporthe oryzae
|
100.0
%
|
|
Journal : Chem Pharm Bull (Tokyo)
Year : 2007
Volume : 55
Issue : 12
First Page : 1755
Last Page : 1757
|
Growth inhibition of Alternaria alternata at 50 ug/ml after 4 days by poisoned food technique
|
Alternaria alternata
|
82.3
%
|
|
Journal : Chem Pharm Bull (Tokyo)
Year : 2007
Volume : 55
Issue : 12
First Page : 1755
Last Page : 1757
|
Growth inhibition of Fusarium graminearum at 500 ug/ml after 4 days by poisoned food technique
|
Fusarium graminearum
|
99.4
%
|
|
Journal : Chem Pharm Bull (Tokyo)
Year : 2007
Volume : 55
Issue : 12
First Page : 1755
Last Page : 1757
|
Growth inhibition of Alternaria alternata at 500 ug/ml after 4 days by poisoned food technique
|
Alternaria alternata
|
100.0
%
|
|
Journal : Chem Pharm Bull (Tokyo)
Year : 2007
Volume : 55
Issue : 12
First Page : 1755
Last Page : 1757
|
Growth inhibition of Fusarium graminearum at 50 ug/ml after 4 days by poisoned food technique
|
Fusarium graminearum
|
38.7
%
|
|
Journal : Chem Pharm Bull (Tokyo)
Year : 2007
Volume : 55
Issue : 12
First Page : 1755
Last Page : 1757
|
Antifungal activity against Fusarium solani assessed as inhibition of mycelium growth after 1 week
|
Fusarium solani
|
38.49
ug.mL-1
|
|
Journal : J Agric Food Chem
Year : 2013
Volume : 61
Issue : 11
First Page : 2789
Last Page : 2795
|
Antifungal activity against Alternaria solani assessed as inhibition of mycelium growth after 1 week
|
Alternaria solani
|
14.03
ug.mL-1
|
|
Journal : J Agric Food Chem
Year : 2013
Volume : 61
Issue : 11
First Page : 2789
Last Page : 2795
|
Antifungal activity against Botryotinia fuckeliana assessed as inhibition of mycelium growth after 1 week
|
Botryotinia fuckeliana
|
8.92
ug.mL-1
|
|
Journal : J Agric Food Chem
Year : 2013
Volume : 61
Issue : 11
First Page : 2789
Last Page : 2795
|
Antifungal activity against Colletotrichum gloeosporioides assessed as inhibition of mycelium growth after 1 week
|
Colletotrichum gloeosporioides
|
100.0
ug.mL-1
|
|
Journal : J Agric Food Chem
Year : 2013
Volume : 61
Issue : 11
First Page : 2789
Last Page : 2795
|
Antifungal activity against Cytospora sp. assessed as inhibition of mycelium growth after 1 week
|
Cytospora
|
100.0
ug.mL-1
|
|
Journal : J Agric Food Chem
Year : 2013
Volume : 61
Issue : 11
First Page : 2789
Last Page : 2795
|
Antifungal activity against Fusarium solani assessed as inhibition of mycelium growth at 100 ug/ml after 1 week
|
Fusarium solani
|
72.45
%
|
|
Journal : J Agric Food Chem
Year : 2013
Volume : 61
Issue : 11
First Page : 2789
Last Page : 2795
|
Antifungal activity against Botryotinia fuckeliana assessed as inhibition of mycelium growth at 100 ug/ml after 1 week
|
Botryotinia fuckeliana
|
100.0
%
|
|
Journal : J Agric Food Chem
Year : 2013
Volume : 61
Issue : 11
First Page : 2789
Last Page : 2795
|
Antifungal activity against Alternaria solani assessed as inhibition of mycelium growth at 100 ug/ml after 1 week
|
Alternaria solani
|
80.3
%
|
|
Journal : J Agric Food Chem
Year : 2013
Volume : 61
Issue : 11
First Page : 2789
Last Page : 2795
|
Antifungal activity against Cytospora sp. assessed as inhibition of mycelium growth at 100 ug/ml after 1 week
|
Cytospora
|
38.94
%
|
|
Journal : J Agric Food Chem
Year : 2013
Volume : 61
Issue : 11
First Page : 2789
Last Page : 2795
|
Antifungal activity against Colletotrichum gloeosporioides assessed as inhibition of mycelium growth at 100 ug/ml after 1 week
|
Colletotrichum gloeosporioides
|
49.21
%
|
|
Journal : J Agric Food Chem
Year : 2013
Volume : 61
Issue : 11
First Page : 2789
Last Page : 2795
