Inhibitory activity against the displacement of Picogreen from fMet-tRNA(fMet) by the aminoglycoside
|
Staphylococcus aureus
|
160.0
nM
|
|
Maximal inhibition against the displacement of Picogreen from fMet-tRNA(fMet) by the aminoglycoside
|
Staphylococcus aureus
|
85.0
%
|
|
Maximal inhibition of the aminoglycoside on Staphylococcus aureus IF-2 binding to fMet-tRNA(fMet)
|
Staphylococcus aureus
|
43.0
%
|
|
Inhibition of purified telomerase of Euplotes aediculatus at 50 uM
|
Euplotes aediculatus
|
0.0
%
|
|
Inhibition of telomerase after assembly using recombinant Tetraymena thermophilia TR and TERT at 50 uM
|
Tetrahymena thermophila
|
0.0
%
|
|
Inhibition of telomerase before assembly using recombinant Tetraymena thermophilia TR and TERT at 50 uM
|
Tetrahymena thermophila
|
0.0
%
|
|
Inhibition of human telomerase before assembly using recombinant hTR and hTERT at 50 uM
|
Homo sapiens
|
25.0
%
|
|
Binding affinity to A-site RNA
|
None
|
50.0
nM
|
|
Cytotoxicity against african green monkey Vero cells after 72 hrs by MTT assay
|
Chlorocebus sabaeus
|
62.5
ug.mL-1
|
|
Antitubercular activity against Mycobacterium tuberculosis H37Rv by BacTiter-Gl Microbial Cell Viability assay
|
Mycobacterium tuberculosis H37Rv
|
70.0
nM
|
|
Antitubercular activity against Mycobacterium tuberculosis H37Rv by microdilution alamar Blue broth assay
|
Mycobacterium tuberculosis H37Rv
|
120.0
nM
|
|
Antimicrobial activity against Mycobacterium tuberculosis H37Rv after 7 days by BacTiter-Glo assay
|
Mycobacterium tuberculosis H37Rv
|
70.0
nM
|
|
Antimycobacterial activity against Mycobacterium tuberculosis H37Rv assessed as growth inhibition by Alamar Blue staining-based broth microdilution assay
|
Mycobacterium tuberculosis H37Rv
|
70.0
nM
|
|
Antimycobacterial activity against Mycobacterium tuberculosis H37Rv ATCC 27294 after 7 days by microplate Alamar blue assay
|
Mycobacterium tuberculosis H37Rv
|
0.07
ug.mL-1
|
|
Antimycobacterial activity against Mycobacterium tuberculosis H37Rv ATCC 27294 at 0.08 ug/ml after 7 days by microplate Alamar blue assay relative to control
|
Mycobacterium tuberculosis H37Rv
|
79.8
%
|
|
Antimycobacterial activity against Mycobacterium tuberculosis H37Rv ATCC 27294 at 0.16 to 0.31 ug/ml after 7 days by microplate Alamar blue assay relative to control
|
Mycobacterium tuberculosis H37Rv
|
96.0
%
|
|
Antimycobacterial activity against Mycobacterium tuberculosis H37Rv ATCC 27294 at 0.63 ug/ml after 7 days by microplate Alamar blue assay relative to control
|
Mycobacterium tuberculosis H37Rv
|
97.3
%
|
|
Antimycobacterial activity against Mycobacterium tuberculosis H37Rv ATCC 27294 at 1.25 to 5 ug/ml after 7 days by microplate Alamar blue assay relative to control
|
Mycobacterium tuberculosis H37Rv
|
98.0
%
|
|
Antimycobacterial activity against Mycobacterium tuberculosis H37Rv assessed as growth inhibition by microdilution AlamarBlue broth assay
|
Mycobacterium tuberculosis H37Rv
|
70.0
nM
|
|
Antimicrobial activity against Mycobacterium tuberculosis H37Rv ATCC 27294 incubated for 7 days by BacTiter-Glo cell viability assay
|
Mycobacterium tuberculosis H37Rv
|
102.0
nM
|
|
Antibacterial activity against Pseudomonas aeruginosa PA7 DSM 24068 after 18 hrs
|
Pseudomonas aeruginosa PA7
|
3.8
ug.mL-1
|
|
Antimicrobial activity against Mycobacterium tuberculosis H37Rv by Alamar blue assay
|
Mycobacterium tuberculosis H37Rv
|
70.0
nM
|
|
Cytotoxicity against monkey Vero cells assessed as decrease in cell viability after 72 hrs by MTT assay
|
Chlorocebus sabaeus
|
6.25
ug.mL-1
|
|
Antimycobacterial activity against Mycobacterium tuberculosis H37Rv
|
Mycobacterium tuberculosis H37Rv
|
80.0
nM
|
|
Binding affinity to 16S rRNA A-site in Escherichia coli S30 extract assessed as inhibition of translation measured after 30 mins by coupled transcription/translation-based luciferase reporter gene assay
|
Escherichia coli
|
70.0
nM
|
|
Antimycobacterial activity against Mycobacterium tuberculosis H37Rv assessed as inhibition of bacterial growth by microdilution alamar blue broth assay
|
Mycobacterium tuberculosis
|
70.0
nM
|
|
Antimycobacterial activity against Mycobacterium tuberculosis H37Rv assessed as inhibition of bacterial growth at 0.17 mM by microdilution alamar blue broth assay relative to control
|
Mycobacterium tuberculosis
|
30.0
%
|
|